What is TRPM2

Transient receptor potential cation channel, subfamily M, member 2, also known as TRPM2, is a human gene.

The protein encoded by this gene is a calcium-permeable cation channel that is regulated by free intracellular ADP-ribose. The encoded protein is activated by oxidative stress and confers susceptibility to cell death. Several alternatively spliced transcript variants of this gene have been described, but their full-length nature is not known.

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Permeability and activation of TRPM

The relative permeability of calcium and magnesium varies widely among TRPM channels. TRPM4/5 are impermeable to calcium. TRPM3/6/7 are highly permeable to both calcium and magnesium. The mechanism of activation also varies greatly among TRPM channels. TRPM2 is activated by ADP-ribose Adenosine 5'-diphosphoribose and functions as a sensor of redox status in cells.[3] TRPM4/5 are activated by intracellular calcium. TRPM8, conversely, can be activated by low temperatures, menthol, eucalyptol and icilin.

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